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Mediation of nitrous oxide analgesia in mice by spinal and supraspinal κ-opioid receptors
Journal article   Peer reviewed

Mediation of nitrous oxide analgesia in mice by spinal and supraspinal κ-opioid receptors

R.M Quock, J.A Best, D.C Chen, L.K Vaughn, P.S Portoghese and A.E Takemori
European journal of pharmacology, Vol.175(1), pp.97-100
1990
Handle:
https://hdl.handle.net/2376/107756
PMID: 2157601

Abstract

Analgesia Nitrous oxide Opioid receptors Narcotic antagonists
Exposure to nitrous oxide produced concentration-dependent analgesia in the mouse abdominal construction test. Intracerebroventricular or intrathecal pretreatment with naltrexone or nor-binaltorphimine significantly reduced nitrous oxide analgesia. However, similar pretreatment with β-funaltrexamine had no appreciable effect. These findings suggest that nitrous oxide analgesia involves spinal and supraspinal κ-opioid receptors.

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